Purpose
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A brain-permeable SIRT2 inhibitor
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Characteristics
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A potent and selective sirtuin 2 deacetylase (SIRT2) inhibitor. Reduces neuronal cholesterol by inhibiting SIRT2 activity.
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Purity
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≥ 98?% by HPLC
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Chemical Name
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3-(1-azepanylsulfonyl)-N-(3-bromphenyl)benzamide
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Formula
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C??H??BrN?O?S
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Permeability
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Cell-permeable
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Solubility
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DMSO
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