Purpose
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GSK1838705A is a potent IGF-1R inhibitor with IC50 of 2.0 nM, modestly potent to IR and ALK with IC50 of 1.6 nM and 0.5 nM, respectively, and little activity to other protein kinases.
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Characteristics
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Target: TGF-beta/Smad inhibitor, IGF-1R inhibitor Receptor: ALK/insulin receptor/IGF-1R/RSK1 Status: Undetermined activity
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Purification
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All the products are sent with COA, HPLC and NMR inspection report to guarantee the quality.
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Purity
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100?%
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Formula
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C27H29FN8O3
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Solubility
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DMSO >107mg/mL, Water <1mg ml="" <="" td="">
1mg> |