Purpose
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BX795 is a potent and specific PDK1 inhibitor with IC50 of 6 nM, 140- and 1600-fold more selective for PDK1 than PKA and PKC in cell-free assays, respectively. Meanwhile, in comparison to GSK3β more than 100-fold selectivity observed for PDK1.
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Characteristics
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Target: PDK inhibitor,c-Kit inhibitor, CDK inhibitor, PKA inhibitor Receptor: PDE1/TBK1,c-kit,CDK2,PKA
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Purification
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All the products are sent with COA, HPLC and NMR inspection report to guarantee the quality.
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Purity
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98?%
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Formula
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C23H26IN7O2S
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Solubility
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DMSO > 100mM
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