Purpose
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PRT062607 (P505-15, BIIB057) HCl is a novel, highly selective Syk inhibitor with IC50 of 1 nM in cell-free assays, >80-fold selective for Syk than Fgr, Lyn, FAK, Pyk2 and Zap70.
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Characteristics
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Target: Syk inhibitor Receptor: Syk,FGR,MLK1,YES,FLT3,PAK5,Lyn,c-Src, LCK Status: experimental
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Purification
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All the products are sent with COA, HPLC and NMR inspection report to guarantee the quality.
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Purity
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97?% +
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Formula
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C19H23N9O.HCl
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Solubility
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200 mM in DMSO and ethanol
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